High-Throughput Screening Products & Reviews

BellBrook Labs’ Lead Discovery Services deliver expert support for hit-to-lead efforts. From inhibitor screening and potency profiling to residence-time, mechanism-of-action, and selectivity studies, their team tailors efficient enzymatic assays to your program—accelerating lead advancement with precision and flexibility.

The Transcreener® cGAMP cGAS Assay Kit offers mix-and-read fluorescent detection of cGAMP—the product of cGAS activity—with no coupling enzymes required. Available in FP or TR‑FRET readouts (far-red tracers minimize interference), it’s HTS-ready (Z’ ≥ 0.7), automation-compatible, and validated on 96‑, 384‑, and 1536‑well formats for enzyme kinetics, SAR, and inhibitor screening.

The CD73 activity assay for HTS and hit-to-lead. Measure specific activity of CD73 in a simple mix-and-read format. The kit is designed for compound library screening and follow-up inhibitor discovery.

The Transcreener dAMP Exonuclease Assay directly measures dAMP produced by exonuclease enzymes as they cleave polynucleotides. 

The Transcreener® GDP GTPase Assay Kit directly measures GDP produced during GTP hydrolysis in a homogeneous mix‑and‑read format—no coupling enzymes needed. Compatible with GTPases, GAPs, and GEFs, it supports FP, FI, and TR‑FRET readouts using far‑red tracers to reduce interference. HTS‑ready with excellent sensitivity (Z′ ≥ 0.7), it streamlines screening and profiling workflows.

Kinetic Plate Imager for reliable and stable high throughput screening

Simplify your omics research

Resolve cross-functional pathways

Prep your samples, dry them on your LazWell plate, stack ‘em in the Luxon and start it. Best part is, there are virtually no false positives when using the LDTD technology, so it’s the perfect alternative to your EIA high-throughput screening methods. Wanna do it even faster? With our Luxon-HTS model, you can go below 1 second per sample. Talk about high-speed analysis!

Results in minutes not hours.

Vapourtec offers a range of world class peptide synthesizer systems offering fast flow solid phase peptide synthesis from 0.05 mmol to 30 mmol.

Highly diverse libraries with 95% guaranteed coverage and industry-leading acceptance rate, delivered in as little as 2 weeks

GenScript's proprietary platforms offer a wide range of ready-to-use peptides, ensuring high-quality, HPLC-purified products for fast, cutting-edge research.

The new standard of excellence in quantitative metabolomics profiling

Our hERG Safety Screening service employs the Synchropatch-384 automated patch clamp system to assess compound effects on the hERG potassium channel. This high-throughput assay detects inhibitors that may prolong QT intervals and cause arrhythmias, aiding early drug safety evaluation. With precise data under physiological conditions, it supports regulatory compliance to advance safer therapeutics. 

Recombinant Human B-cell Maturation Antigen (BCMA/TNFRSF17), a TNF receptor superfamily member that is a clinically validated target for multiple myeloma therapies.

Unraveling the complexity of disease

Transforming medicine with metabolomics

Gyrolab® Bioaffy™ 4000, the newest member of the Gyrolab Bioaffy family, offers 2-6 fold extended sensitivity for PK and biomarker analysis compared to Gyrolab Bioaffy 1000.

Decoding lipid-driven biology

As part of Roche’s NGS Automation solutions, AVENIO Edge System is a fully automated system for library preparation, target enrichment, pooling, normalization, and quantification. AVENIO Edge System is designed to simplify the complexity of automation and optimize lab resources, providing the freedom to walk away and work away, with confidence and trust.

Efficient workflows for busy laboratories

KCGS is a comprehensive collection of 295 highly selective kinase inhibitors targeting 262 human kinases

Highly diverse libraries with 95% guaranteed coverage and industry-leading acceptance rate, delivered in as little as 2 weeks.